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Mutant IDH1 inhibitor

CAS No. 1429180-08-4

Mutant IDH1 inhibitor ( —— )

产品货号. M23590 CAS No. 1429180-08-4

Mutant IDH1 inhibitor is an effective inhibitor of mutant IDH1 R132H (IC50: < 72 nM).

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥1361 有现货
10MG ¥2333 有现货
25MG ¥3929 有现货
50MG ¥5613 有现货
100MG ¥7995 有现货
500MG ¥15957 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Mutant IDH1 inhibitor
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Mutant IDH1 inhibitor is an effective inhibitor of mutant IDH1 R132H (IC50: < 72 nM).
  • 产品描述
    Mutant IDH1 inhibitor is an effective inhibitor of mutant IDH1 R132H (IC50: < 72 nM).
  • 同义词
    ——
  • 通路
    Metabolic Enzyme/Protease
  • 靶点
    Dehydrogenase
  • 受体
    mutant IDH1 R132H
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    1429180-08-4
  • 分子量
    466.6
  • 分子式
    C25H34N6O3
  • 纯度
    >98% (HPLC)
  • 溶解度
    DMSO:30 mg/mL (64.3 mM)
  • SMILES
    CC(C)[C@@H](COC1=O)N1c1nc(N[C@@H](C)c2ccc(CN(CC3)CCN3C(C)=O)cc2)ncc1
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.3-Pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant IDH and their preparation. Patent WO 2013046136 A1 20130404
产品手册
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